1149362-69-5Relevant academic research and scientific papers
[2-(4-Phenyl-4-piperidinyl)ethyl]amine based CCR5 antagonists: derivatizations at the N-terminal of the piperidine ring
Duan, Maosheng,Aquino, Christopher,Ferris, Robert,Kazmierski, Wieslaw M.,Kenakin, Terry,Koble, Cecilia,Wheelan, Pat,Watson, Chris,Youngman, Michael
scheme or table, p. 1610 - 1613 (2009/11/30)
Several series of CCR5 antagonists have been discovered by derivatization at the N-terminal of the piperidine ring of the core template 2. Some derivatives exhibited potent inhibition against HIV-1infection. The pharmacokinetic properties of the lead comp
