1150542-85-0Relevant articles and documents
AZAINDOLE DERIVATIVES
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Page/Page column 37, (2011/09/16)
Compounds of the formula (I), in which X1, X2, X3, X4, R1, R2, R3 and R4 have the meanings indicated in Claim 1, are inhibitors of tyrosine kinases, in particular Met
Syntheses of novel 2,3-diaryl-substituted 5-cyano-4-azaindoles exhibiting c-Met inhibition activity
Koolman, Hannes,Heinrich, Timo,Boettcher, Henning,Rautenberg, Wilfried,Reggelin, Michael
scheme or table, p. 1879 - 1882 (2009/11/30)
Herein we report the syntheses of 2,3-diaryl-substituted pyrrolo[3,2-b]pyridine-5-carbonitriles via a one-pot 5-endo-dig-cyclization/protection reaction followed by palladium catalyzed arylation. In addition, a complementary synthesis route employing Laro