115201-07-5Relevant articles and documents
Highly diastereo- and enantioselective aziridination of α,β-unsaturated amides with diaziridine and mechanistic consideration on its stereochemistry
Ishihara, Hiroyuki,Hori, Kiyoto,Sugihara, Hiroyasu,Ito, Yoshio N.,Katsuki, Tsutomu
, p. 4272 - 4286 (2007/10/03)
During studies of aziridination of α,β-unsaturated amides with diaziridine, we found that we could prepare both the cis- and trans-aziridinecarboxamides by choosing an appropriately substituted diaziridine. While 3-monosubstituted diaziridine 2 was suitab