1161743-52-7Relevant articles and documents
1-Alkyl-8-(piperazine-1-sulfonyl)phenylxanthines: Development and characterization of adenosine A2B receptor antagonists and a new radioligand with subnanomolar affinity and subtype specificity
Borrmann, Thomas,Hinz, Sonja,Bertarelli, Daniela C. G.,Li, Wenjin,Florin, Nicole C.,Scheiff, Anja B.,Müller, Christa E.
experimental part, p. 3994 - 4006 (2010/01/06)
A new series of 1-alkyl-8-(piperazine-1-sulfonyl)phenylxanthines was designed, synthesized, and characterized in radioligand binding and functional assays at A2B adenosine receptors. A2B antagonists with subnanomolar affinity and hig