1164273-86-2Relevant academic research and scientific papers
PENICILLIN-BINDING PROTEIN INHIBITORS
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Paragraph 00174, (2021/06/04)
Described herein are certain boron-containing compounds, compositions, preparations and their use as modulators of the transpeptidase function of bacterial penicillin-binding proteins and as antibacterial agents. In some embodiments, the compounds describ
PENICILLIN-BINDING PROTEIN INHIBITORS
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Paragraph 00357, (2019/12/15)
Described herein are certain boron-containing compounds, compositions, preparations and their use as modulators of the transpeptidase function of bacterial penicillin-binding proteins and as antibacterial agents. In some embodiments, the compounds describ
Synthesis and evaluation of radamide analogues, a chimera of radicicol and geldanamycin
Hadden, M. Kyle,Blagg, Brian S. J.
supporting information; experimental part, p. 4697 - 4704 (2009/10/17)
(Chemical Equation Presented) Previously, we reported the Hsp90 inhibitory activity of radamide, an open chain amide chimera of geldanamycin and radicicol. Attempts to further expand upon structure-activity relationships for this class of Hsp90 inhibitors
