1170675-32-7Relevant academic research and scientific papers
Identification of peptide substrate and small molecule inhibitors of Testis-Specific Serine/Threonine Kinase1 (TSSK1) by the developed assays
Zhang, Leilei,Yan, Yu,Liu, Zijie,Abliz, Zeper,Liu, Gang
experimental part, p. 4419 - 4428 (2010/03/01)
In this paper, a peptide substrate (Pep8) of TSSK1 is identified. Using Pep8 as a substrate, two homogeneous and efficient assays for TSSK1 inhibitors screening have been developed, including luminescent kinase assay and LC-MS-based high-throughput assay.
