1173103-85-9Relevant articles and documents
2-Substituted 5,6-dimethyl-3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidines: New series of highly potent and specific serotonin 5-HT6 receptor antagonists
Ivachtchenko, Alexandre V.,Golovina, Elena S.,Kadieva, Madina G.,Koryakova, Angela G.,Mitkin, Oleg D.,Tkachenko, Sergey E.,Kysil, Volodymyr M.,Okun, Ilya
, p. 1189 - 1197 (2011)
Syntheses, biological evaluation, and structure-activity relationships for a series of novel 2-substituted 3-benzenesulfonyl-5,6-dimethyl-pyrazolo[1,5-a] pyrimidines are disclosed. In spite of a wide, four orders of magnitude, SAR range (Ki var