1174730-89-2Relevant academic research and scientific papers
Hit-to-lead optimization of pyrrolo[1,2-a]quinoxalines as novel cannabinoid type 1 receptor antagonists
Szabo, Gyoergy,Kiss, Robert,Payer-Lengyel, Dora,Vukics, Krisztina,Szikra, Judit,Baki, Andrea,Molnar, Laszlo,Fischer, Janos,Keseru, Gyoergy M.
scheme or table, p. 3471 - 3475 (2010/02/28)
Hit-to-lead optimization of a novel series of N-alkyl-N-[2-oxo-2-(4-aryl-4H-pyrrolo[1,2-a]quinoxaline-5-yl)-ethyl]-car boxylic acid amides, derived from a high throughput screening (HTS) hit, are described. Subsequent optimization led to identification of
