1180007-72-0Relevant articles and documents
Pd(II)-catalyzed o-C-H acetoxylation of phenylalanine and ephedrine derivatives with MeCOOOtBu/Ac2O
Vickers, Chris J.,Mei, Tian-Sheng,Yu, Jin-Quan
supporting information; experimental part, p. 2511 - 2513 (2010/07/06)
Pd(II)-catalyzed ortho C-H acetoxylation of triflate protected phenethyl- and phenpropylamines has been achieved with tert-butyl peroxyacetate as the stoichiometric oxidant and either DMF or CH3CN as the promoter. The reaction was found to tolerate a large variety of functional groups and could be combined with subsequent intramolecular amination to afford functionalized indoline derivatives.