1192234-98-2Relevant academic research and scientific papers
Novel 2H-isoquinolin-3-ones as antiplasmodial falcipain-2 inhibitors
Micale, Nicola,Ettari, Roberta,Schirmeister, Tanja,Evers, Astrid,Gelhaus, Christoph,Leippe, Matthias,Zappala, Maria,Grasso, Silvana
experimental part, p. 6505 - 6511 (2009/12/06)
A series of 1-aryl-6,7-disubstituted-2H-isoquinolin-3-ones (2-10) was synthesized and evaluated for their inhibition against Plasmodium falciparum cysteine protease falcipain-2, as well as against cultured P. falciparum strain FCBR parasites. All compound
