1195785-11-5Relevant articles and documents
Synthesis and biological activities of 4-substituted pyrrolo[2,3-a] carbazole Pim kinase inhibitors
Giraud, Francis,Akué-Gédu, Rufine,Nauton, Lionel,Candelon, Nicolas,Debiton, Eric,Théry, Vincent,Anizon, Fabrice,Moreau, Pascale
, p. 225 - 236 (2013/01/15)
Pyrrolo[2,3-a]carbazole-3-carbaldehydes are potent Pim kinase inhibitors with in vitro antiproliferative activities. In the present study, we report the synthesis and biological activities (Pim kinase inhibition and in vitro antiproliferative potency) of