1196066-46-2Relevant academic research and scientific papers
Synthesis and biological evaluation of 2-alkynyl-N6-methyl- 5′-N-methylcarboxamidoadenosine derivatives as potent and highly selective agonists for the human adenosine A3 receptor
Volpini, Rosaria,Buccioni, Michela,Dal Ben, Diego,Lambertucci, Catia,Lammi, Carmen,Marucci, Gabriella,Ramadori, Anna T.,Klotz, Karl-Norbert,Cristalli, Gloria
experimental part, p. 7897 - 7900 (2010/06/12)
A new series of 2-aralkynyl-N6-methyl-MECAs 10-13 were synthesized and evaluated in radioligand binding studies and in a newEu-GTP functional assay that provides a powerful alternative to radioisotope use. The new compounds possess high affinit
