119730-33-5Relevant academic research and scientific papers
5 H - thiazolo [3, 2 - a] pyrimidine - 5 - ketone derivative and its preparation method and used as antibacterial medicament application
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Paragraph 0039; 0100-0102, (2017/08/23)
The invention discloses 5H-thiazolo[3,2-a]pyrimidyl-5-one derivatives which have a definite chemical structure and are simple in chemical structure. The invention also discloses a preparation method of the 5H-thiazolo[3,2-a]pyrimidyl-5-one derivatives, wh
Synthesis of some new thiazolo[3,2-A]pyrimidine derivatives and screening of their in vitro antibacterial and antitubercular activities
Cai, Dong,Zhang, Zhi-Hua,Chen, Yu,Yan, Xin-Jia,Zhang, Shi-Ti,Zou, Liang-Jing,Meng, Li-Hong,Li, Fang,Fu, Bing-Jie
, p. 292 - 302 (2016/01/25)
The novel 5H-thiazolo[3,2-A]pyrimidin-5-ones were synthesized by thiophene ring closure. The first step is the synthesis of S-alkylated derivatives by the reaction of 6-substituted-2-thiouracils with the appropriate substituted phenacyl halides. Upon trea
The Chemistry of Pyrimidinethiols. II. The Preparation and Reaction of Some 2-Arenecarbonylmethylthiopyrimidines
Hurst, Derek T.,Beaumont, Claire,Jones, Derek T. E.,Kingsley, Deborah A.,Partridge, Julian D.,Rutherford, Trevor J.
, p. 1209 - 1219 (2007/10/02)
A number of 2-arenecarbonylmethylthiopyrimidin-4(1H)-ones has been synthesized.Those having H, Me or Pr as a 6-substituent undergo ready sulfur extrusion on heating in diphenyl ether to give 2-(arenecarbonylmethylene)-2,3-dihydropyrimidin-4(1H)-ones, but
