1202252-05-8Relevant academic research and scientific papers
BENZO[d]OXAZOLES AND BENZO[d]THIAZOLES AS KINASE INHIBITORS
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Page/Page column 83-84, (2010/04/06)
Novel benzo[d]oxazole and/or benzo[d]thiazole compounds, pharmaceutical compositions containing the benzo[d]oxazole and/or benzo[d]thiazole compounds, and methods of their pharmaceutical use are disclosed. In certain embodiments, the benzo[d]oxazole and/o
Benzothiazoles as Rho-associated kinase (ROCK-II) inhibitors
Yin, Yan,Lin, Li,Ruiz, Claudia,Cameron, Michael D.,Pocas, Jennifer,Grant, Wayne,Schroeter, Thomas,Chen, Weimin,Duckett, Derek,Schuerer, Stephan,LoGrasso, Philip,Feng, Yangbo
scheme or table, p. 6686 - 6690 (2010/06/14)
A series of benzothiazole derivatives as ROCK inhibitors have been discovered. Compounds with good biochemical and cellular potency, and sufficient kinase selectivity have been identified.
