1202483-45-1Relevant articles and documents
2-Amino-[1,2,4]triazolo[1,5-a]pyridines as JAK2 inhibitors
Siu, Michael,Pastor, Richard,Liu, Wendy,Barrett, Kathy,Berry, Megan,Blair, Wade S.,Chang, Christine,Chen, Jacob Z.,Eigenbrot, Charles,Ghilardi, Nico,Gibbons, Paul,He, Haiying,Hurley, Christopher A.,Kenny, Jane R.,Cyrus Khojasteh,Le, Hoa,Lee, Leslie,Lyssikatos, Joseph P.,Magnuson, Steve,Pulk, Rebecca,Tsui, Vickie,Ultsch, Mark,Xiao, Yisong,Zhu, Bing-Yan,Sampath, Deepak
, p. 5014 - 5021 (2013/09/02)
The advancement of a series of ligand efficient 2-amino-[1,2,4]triazolo[1, 5-a]pyridines, initially identified from high-throughput screening, to a JAK2 inhibitor with pharmacodynamic activity in a mouse xenograft model is disclosed.