1204403-89-3Relevant academic research and scientific papers
Evaluation of (4-Arylpiperidin-1-yl)cyclopentanecarboxamides As High-Affinity and Long-Residence-Time Antagonists for the CCR2 Receptor
Vilums, Maris,Zweemer, Annelien J. M.,Dilanchian, Arian,Vanveldhoven, Jacobus P. D.,Devries, Henk,Brussee, Johannes,Saunders, John,Stamos, Dean,Heitman, Laura H.,Ijzerman, Adriaan P.
, p. 1249 - 1258 (2015)
Animal models suggest that the chemokine ligand 2/CC-chemokine receptor 2 (CCL2/CCR2) axis plays an important role in the development of inflammatory diseases. However, CCR2 antagonists have failed in clinical trials because of a lack of efficacy. We prev
