1211284-05-7Relevant articles and documents
Highly functional group compatible Rh-catalyzed addition of arylboroxines to activated N-tert-butanesulfinyl ketimines
Jung, Hyung Hoon,Buesking, Andrew W.,Ellman, Jonathan A.
supporting information; experimental part, p. 3912 - 3915 (2011/09/16)
The rhodium-catalyzed addition of readily accessible arylboroxines to N-tert-butanesulfinyl ketimines derived from oxetan-3-one, N-Boc-azetidin-3-one, and isatins proceeds in high yields with excellent functional group compatibility. Moreover, high diastereoselectivities are observed for the additions to the N-sulfinyl ketimines derived from isatins.
Reactions of oxetan-3-tert-butylsulfinimine for the preparation of substituted 3-aminooxetanes
Hamzik, Philip J.,Brubaker, Jason D.
supporting information; experimental part, p. 1116 - 1119 (2010/06/11)
(Figure Presented) The oxetane ring Is useful In drug discovery as a bioisostere for both the geminal dimethyl group and the carbonyl group. A convenient, straightforward approach to access structurally diverse 3-aminooxetanes through the reactivity of oxetan-3-tert-butylsulfinimine and the corresponding sulfinylaziridine Is described.