1213786-08-3Relevant academic research and scientific papers
Metal-free synthesis of 3-sulfenylindoles via an iodine-mediated electrophilic cyclisation of 2-alkynylanilines with disulfides
Tao, Li-Ming,Liu, Wen-Qi,Zhou, Yun,Li, Ai-Tao
, p. 644 - 646 (2012)
An efficient and metal-free method was developed to synthesise 3-sulfenylindoles via the iodine-mediated electrophilic cyclisation of 2-alkynylanilines with disulfides. In the presence of I2, various 3-sulfenylindoles were obtained in moderate
Palladium-catalyzed annulation of 2-(1-Alkynyl)benzenamines with disulfides: Synthesis of 3-sulfenylindoles
Guo, Yan-Jin,Tang, Ri-Yuan,Li, Jin-Heng,Zhong, Ping,Zhang, Xing-Guo
supporting information; experimental part, p. 2615 - 2618 (2009/12/29)
3-Sulfenylindoles can be efficiently prepared in moderate to good yields from 2-(1-alkynyl)benzenamines and disulfides using the palladium/air catalytic systems. The study also provides a useful route to the synthesis of fipronil analogues.
