121806-83-5

Upstream product

• 262855-60-7 tert-butyl 2-[(2-{bis[2-(tert-butoxy)-2-oxoethyl]amino}-3-(4-nitrophenyl)propyl)(2-{bis[2-(tert-butoxy)-2-oxoethyl]amino}ethyl)amino]acetate 
• 463-71-8 thiophosgene 
• 128817-52-7 2-{[3-(4-aminophenyl)-2-[bis(carboxymethyl)amino]propyl] ({2-[bis(carboxymethyl)amino]ethyl})amino}acetic acid 

Downstream Products

• 620609-93-0 N-[(2,3,4,5,6-pentafluorophenyl)carboxamide-]-N-[2-(4-{[(cyclohexylamino)carbonyl]amino}sulfonyl)ethyl]-2-p-phenylmethyl(diethylenetriamine-N,N,N',N'',N''-pentaacetic acid) 
• 1034685-17-0 2-{N-[8-(3-trifluoromethyl-7-oxabicyclo[2.2.1]hepta-2,5-dien-2-ylcarbonyl)-3,6-dioxaoct-1-yl]thioureidobenzyl}diethylenetriaminepentaacetic acid 
• 1263049-49-5 N-(2-[bis(carboxymethyl)amino]-3-{4-[(dodecylcarbamothioyl)amino]phenyl}propyl)-N-{2-[bis(carboxymethyl)amino]ethyl}glycine 
• 1263049-50-8 12-{[(4-{2-[bis(carboxymethyl)amino]-3-[{2-[bis(carboxymethyl)amino]ethyl}(carboxymethyl)amino]propyl}phenyl)carbamothioyl]amino}dodecanoic acid 
• 1559003-54-1 C₃₈H₅₈N₈O₁₄S₂ 

Relevant academic research and scientific papers

SYNTHESIS OF THERAPEUTIC AND DIAGNOSTIC DRUGS CENTERED ON REGIOSELECTIVE AND STEREOSELECTIVE RING OPENING OF AZIRIDINIUM IONS

Stereoselective and regioselective synthesis of compounds via nucleophilic ring opening reactions of aziridinium ions for use in stereoselective and regioselective synthesis of therapeutic and diagnostic compounds.

Backbone polysubstituted chelates for forming a metal chelate-protein conjugate

New polysubstituted diethylenetriaminepentaacetic acid chelates and protein conjugates of the same are described together with the methods of preparing such compounds. A method of delivering radiolabelled compound of the present invention to a target site while minimizing the distribution of the compound to non-targeted organs or tissues is also disclosed.