1220219-22-6Relevant articles and documents
Radical Metal-Free Borylation of Aryl Iodides
Pinet, Sandra,Liautard, Virginie,Debiais, Mégane,Pucheault, Mathieu
, p. 4759 - 4768 (2017/10/03)
A simple metal-free borylation of aryl iodides mediated by a fluoride sp 2 -sp 3 diboron adduct is described. The reaction conditions are compatible with various functional groups. Electronic effects of substituents do not affect the borylation while steric hindrance does. The reaction proceeds via a radical mechanism in which pyridine serves to stabilize the boryl radicals, generated in situ.
COMPOSITIONS AND THERAPEUTIC USES OF IKK-RELATED KINASE EPSILON AND TANKBINDING KINASE 1 INHIBITORS
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Page/Page column 60, (2012/11/06)
The invention relates to compounds, pharmaceutical compositions and medicaments comprising such compounds, and the use of these compounds, compositions, and medicaments in methods of treating diseases and disorders.