1221267-34-0Relevant articles and documents
Pyrrolo[1,2-f]triazines as JAK2 inhibitors: Achieving potency and selectivity for JAK2 over JAK3
Harikrishnan, Lalgudi S.,Kamau, Muthoni G.,Wan, Honghe,Inghrim, Jennifer A.,Zimmermann, Kurt,Sang, Xiaopeng,Mastalerz, Harold A.,Johnson, Walter L.,Zhang, Guifen,Lombardo, Louis J.,Poss, Michael A.,Trainor, George L.,Tokarski, John S.,Lorenzi, Matthew V.,You, Dan,Gottardis, Marco M.,Baldwin, Kathy F.,Lippy, Jonathan,Nirschl, David S.,Qiu, Ruhui,Miller, Arthur V.,Khan, Javed,Sack, John S.,Purandare, Ashok V.
, p. 1425 - 1428 (2011/04/16)
SAR studies of pyrrolo[1,2-f]triazines as JAK2 inhibitors is presented. Achieving JAK2 inhibition selectively over JAK3 is discussed.