1224947-47-0Relevant articles and documents
Synthesis of 5-Aryl- and 5-Heteroaryl-7-carboxyl-8-hydroxyquinaldines through Suzuki cross-coupling reaction with potassium organotrifluoroborates
Sliman, Faten,Desmaele, Didier
experimental part, p. 619 - 630 (2010/04/26)
A series of 5-aryl- and 5-heteroaryl-7-carboxyl-8-hydroxyquinaldines were prepared from 5-bromo-7-methoxycarbonyl-8-benzyloxyquinaldine based on the Suzuki cross-coupling reaction using potassium organotrifluoroborates. An efficient method of deprotection of the 8-hydroxy group using a microwave-assisted hydrogen transfer reaction is reported. Georg Thieme Verlag Stuttgart · New York.