1228083-47-3Relevant academic research and scientific papers
Proteasome selectivity towards Michael acceptor containing oligopeptide-based inhibitors
Van Der Linden, Wouter A.,Geurink, Paul P.,Oskam, Chris,Van Der Marel, Gijsbert A.,Florea, Bogdan I.,Overkleeft, Herman S.
, p. 1885 - 1893 (2010)
The synthesis and biological evaluation of ten Michael acceptors containing potential proteasome inhibitors are described. Cellular targets of azide containing inhibitors Ib and VIIIb were assessed in HEK293T and RAW264.7 cells by a two step labeling stra
