1233504-67-0Relevant academic research and scientific papers
Discovery of a novel series of nonsteroidal androgen receptor modulators: 5- or 6-oxachrysen-2-ones
Zhao, Shuo,Shen, Yixing,van Oeveren, Arjan,Marschke, Keith B.,Zhi, Lin
, p. 3431 - 3435 (2008)
A novel oxachrysenone series (2) of nonsteroidal selective androgen receptor modulators (SARM) was developed based on the 6-aryl-2-quinolinones (1). Synthesis and preliminary SAR results based on in vitro assays are discussed. In the cotransfection assay,
ANDROGEN RECEPTOR MODULATOR COMPOUNDS AND METHODS
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Page/Page column 123, (2008/06/13)
Provided herein are compounds that bind to androgen receptors and/or modulate activity of androgen receptors and/or modulate the amount of androgen receptors; and to methods for making and using such compounds. Also provided are compositions containing su
