124027-46-9Relevant articles and documents
Diazacycloalkyl-1,2,4-triazolo[2,3-c][1,3]benzodiazepines useful as neuroleptic and/or antihistaminic agents
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, (2008/06/13)
Described are 5-diazacycloalkyltriazolo[2,3-c][1,3]benzodiazepines, for example compounds of the formula STR1 wherein R1 represents hydrogen, halogen, trifluoromethyl, lower alkylthio, lower alkoxy or lower alkyl; R2 represents hydrogen, lower alkyl or hydroxy-C2 -C7 alkyl wherein the hydroxy group is separated from the nitrogen atom by at least 2 carbon atoms; R3 represents hydrogen, lower alkyl, lower alkoxy, lower alkylthio, halogen or trifluoromethyl; and Cn H2n represents ethylene. The synthesis, pharmaceutical compositions and methods of use as neuroleptic and/or antihistaminic agents are given.