1245834-05-2Relevant academic research and scientific papers
Piperidinyl-nicotinamides as potent and selective somatostatin receptor subtype 5 antagonists
Alker, Andre,Binggeli, Alfred,Christ, Andreas D.,Green, Luke,Maerki, Hans Peter,Martin, Rainer E.,Mohr, Peter
scheme or table, p. 4521 - 4525 (2010/11/24)
Nicotinamides of benzyl-substituted 4-aminopiperidines and their seven-membered analogs of generic structure 2 and 2′ have been discovered as potent and selective SST5 antagonists. The activity (Ki) ranges from 2.4 to 436 nM. Most compounds exh
