1245907-05-4Relevant academic research and scientific papers
3-Cyano-6-(5-methyl-3-pyrazoloamino)pyridines: Selective Aurora A kinase inhibitors
Ando, Ryoichi,Ikegami, Hiroshi,Sakiyama, Makoto,Ooike, Shinsuke,Hayashi, Masayuki,Fujino, Yasuhiro,Abe, Daisuke,Nakamura, Hideo,Mishina, Tadashi,Kato, Harutoshi,Iwase, Yumiko,Tomozane, Hideo,Morioka, Masahiko
, p. 4709 - 4711 (2010)
A new class of Aurora A kinase inhibitor was created by transforming 4-(5-methyl-3-pyrazoloamino)pyrimidine moiety of VX-680 to 3-cyano-6-(5-methyl- 3pyrazoloamino)pyridine. Compound 6 exhibited a potent Aurora A kinase inhibitory activity, excellent selectivity to Aurora B kinase and other 60 kinases, good cell permeability and good PK profile. Therefore compound 6 was effective in antitumor mice model at a dose of 30 mg/kg po qd without decrease of body weight.
