1252672-69-7Relevant articles and documents
Site-Selective Late-Stage Aromatic [18F]Fluorination via Aryl Sulfonium Salts
Xu, Peng,Zhao, Da,Berger, Florian,Hamad, Aboubakr,Rickmeier, Jens,Petzold, Roland,Kondratiuk, Mykhailo,Bohdan, Kostiantyn,Ritter, Tobias
supporting information, p. 1956 - 1960 (2019/12/24)
Site-selective functionalization of C?H bonds in small complex molecules is a long-standing challenge in organic chemistry. Herein, we report a broadly applicable and site-selective aromatic C?H dibenzothiophenylation reaction. The conceptual advantage of this transformation is further demonstrated through the two-step C?H [18F]fluorination of a series of marketed small-molecule drugs.
NOVEL AMIDE AND AMIDINE DERIVATIVES AND USES THEREOF
-
Page/Page column 47, (2010/11/03)
The present invention relates to inhibitors of 11-β-hydroxysteroid dehydrogenase type 1 enzyme and their use in treatment of non-insulin dependent type 2 diabetes, insulin resistance, obesity, lipid disorders, metabolic syndrome, central nervous system disorders, and diseases and conditions that are related to excessive glucocorticoids.