1255305-48-6Relevant articles and documents
Discovery of a novel azetidine scaffold for colony stimulating factor-1 receptor (CSF-1R) Type II inhibitors by the use of docking models
Ikegashira, Kazutaka,Ikenogami, Taku,Yamasaki, Takayuki,Hase, Yasunori,Yamaguchi, Takayuki,Inagaki, Koji,Doi, Satoki,Adachi, Tsuyoshi,Koga, Yoshihisa,Hashimoto, Hiromasa
supporting information, p. 115 - 118 (2018/11/23)
We report the discovery of a novel azetidine scaffold for colony stimulating factor-1 receptor (CSF-1R) Type II inhibitors by using a structure-based drug design (SBDD) based on a docking model. The work leads to the representative compound 4a with high C