1255949-85-9Relevant academic research and scientific papers
Practical and scalable synthesis of a selective CCK1 receptor antagonist
Mapes, Christopher M.,Mani, Neelakandha S.,Deng, Xiaohu,Pandit, Chennagiri R.,McClure, Kelly J.,Pippel, Marna C. W.,Sehon, Clark A.,Gomez, Laurent,Shinde, Shirin,Breitenbucher, J. Guy,Jones, Todd K.
scheme or table, p. 7950 - 7953 (2011/02/22)
We describe a practical and scalable route to compound (Z)-1, a selective CCK1 receptor antagonist. Notable features of this concise route are (1) a regioselective construction of the pyrazole core through the reaction of an aryl hydrazine and
