1261736-75-7Relevant academic research and scientific papers
A borylative cyclisation towards indole boronic esters
Huang, Jianhui,MacDonald, Simon J.F.,Harrity, Joseph P.A.
supporting information; experimental part, p. 8770 - 8772 (2011/02/24)
2-Alkynylaniline borylative cyclisations provide a direct means to access indole 3-boronic esters from simple precursors. The Pd-catalysed cyclisation can be merged with cross-coupling processes in the same reaction vessel, moreover, the products can be e
