1265900-84-2Relevant academic research and scientific papers
Stereospecific synthesis and structure-activity relationships of unsymmetrical 4,4-diphenylbut-3-enyl derivatives of nipecotic acid as GAT-1 inhibitors
Pizzi, Domenica A.,Leslie, Colin P.,Fabio, Romano Di,Seri, Catia,Bernasconi, Giovanni,Squaglia, Michela,Carnevale, Gennaro,Falchi, Alessandro,Greco, Elisabetta,Mangiarini, Laura,Negri, Michele
, p. 602 - 605 (2011)
Two complementary stereospecific synthetic approaches for the preparation of unsymmetrical ortho-substituted N-(4,4-diphenylbut-3-enyl) derivatives of nipecotic acid are described. Determination of the activity of the prepared compounds at the GAT-1 trans
