1272672-03-3Relevant academic research and scientific papers
Discovery of pyridones as oral AMPK direct activators
Mirguet, Olivier,Sautet, Stephane,Clement, Catherine-Anne,Toum, Jeroime,Donche, Frederic,Marques, Celine,Rondet, Emilie,Pizzonero, Mathieu,Beaufils, Benjamin,Dudit, Yann,Huet, Pascal,Trottet, Lionel,Grondin, Pascal,Brusq, Jean-Marie,Boursier, Eric,Saintillan, Yannick,Nicodeme, Edwige
, p. 632 - 636 (2013/07/26)
AMP-activated protein kinase (AMPK) is an evolutionarily conserved fuel-sensing enzyme that is activated in shortage of energy and suppressed in its surfeit. AMPK activation stimulates fatty acid oxidation, enhances insulin sensitivity, alleviates hypergl
PYRROLO-PYRIDINE DERIVATIVES AS ACTIVATORS OF AMPK
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, (2011/04/18)
The present invention relates to pyrrolopyridone compounds of the formula (I), salts thereof, to pharmaceutical compositions containing them and their use in medicine. In particular, the invention relates to compounds as activators of AMPK.
