127625-30-3Relevant articles and documents
Naphthosultam Derivatives: A New Class of Potent and Selective 5-HT2 Antagonists
Malleron, Jean-Luc,Comte, Marie-Therese,Gueremy, Claude,Peyronel, Jean Francois,Truchon, Alain,et al.
, p. 2477 - 2483 (2007/10/02)
A series of 2-(aminoalkyl)naphthisothiazole 1,1-dioxides was synthesized and examined in various receptor binding tests.Most compounds demonstrated high affinity for the 5-HT2 receptor with moderate to high selectivity.A member of this