1286716-55-9Relevant academic research and scientific papers
A convenient synthesis of amino acid arylamides utilizing methanesulfonyl chloride and N-methylimidazole
Mao, Liguang,Wang, Zhenyu,Li, Yongjia,Han, Xiqian,Zhou, Weicheng
supporting information; experimental part, p. 129 - 133 (2011/03/22)
N-Cbz-protected amino acids reacted with various aryl-amines in the presence of methanesulfonyl chloride and N-methylimidazole in dichloromethane to give the corresponding arylamides in high yields. No obvious racemization was observed under the mild conditions. Georg Thieme Verlag Stuttgart - New York.
