1290145-05-9Relevant academic research and scientific papers
Discovery of benzothiazole-based adenosine A2B receptor antagonists with improved A2A selectivity
Firooznia, Fariborz,Cheung, Adrian Wai-Hing,Brinkman, John,Grimsby, Joseph,Gubler, Mary Lou,Hamid, Rachid,Marcopulos, Nicholas,Ramsey, Gwendolyn,Tan, Jenny,Wen, Yang,Sarabu, Ramakanth
, p. 1933 - 1936 (2011/04/24)
The highly potent but modestly selective N-(2-amino-4-methoxy-benzothiazol- 7-yl)-N-ethyl-acetamide derivative 2 was selected as the starting point for the design of novel selective A2B antagonists, due to its excellent potency, and good drug-l
