1292783-99-3Relevant academic research and scientific papers
Spacer Effects on in vivo Properties of DOTA-Conjugated Dimeric [Tyr3]Octreotate Peptides Synthesized by a "CuI-Click" and "Sulfo-Click" Ligation Method
Yim, Cheng-Bin,van der Wildt, Berend,Dijkgraaf, Ingrid,Joosten, Lieke,Eek, Annemarie,Versluis, Cees,Rijkers, Dirk T. S.,Boerman, Otto C.,Liskamp, Rob M. J.
experimental part, p. 750 - 760 (2012/02/01)
We report on the SSTR2-binding properties of a series of four dimeric [Tyr3]octreotate analogues with different spacer lengths (nine, 19, 41, and 57 atoms) between the peptides. Two analogues (9 and 57 atoms) were selected as precursors for the design, sy
