1297529-86-2Relevant academic research and scientific papers
Synthesis and biological evaluation of dibenz[b,f][1,5]oxazocine derivatives for agonist activity at κ-opioid receptor
Mitra, Sudipta,Banerjee, Tuhin Suvro,Hota, Sandip K.,Bhattacharya, Debleena,Das, Sumantra,Chattopadhyay, Partha
, p. 1713 - 1720 (2011/05/06)
A short and high yield synthetic route to dibenz[b,f][1,5]oxazocines has been developed using Pd catalyzed intramolecular cycloamination reaction. Receptor binding assay using [125I]-dynorphin demonstrated that one of the derivative, 5b showed
