1306739-68-3Relevant articles and documents
Preparation method and intermediate of heteroaryl [4, 3-c] pyrimidine-5-amine compound
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Paragraph 0110-0112, (2020/11/12)
The invention relates to a preparation method and an intermediate of a heteroaryl [4, 3-c] pyrimidine-5-amine compound. Specifically, the present invention relates to a heteroaryl [4, 3-c] pyrimidine-5-amine compound or a preparation method of its salt. The method comprises the following steps: preparing a compound as shown in a formula II from a compound as shown in a formula III, and reacting the compound as shown in the formula II serving as a raw material to obtain a compound as shown in a formula I. In the reaction process, few impurities are generated, the purification process is simplified, and the preparation method is suitable for industrialization.