1307296-47-4

Upstream product

• 4972-29-6 benzenesulphinyl chloride 
• 38235-77-7 (R)-N-benzyl-1-phenylethylamine 
• 1307296-48-5 (R,S)-N-Benzyl-N-(1-phenylethyl)-p-toluenesulfinamide 
• 1307296-49-6 (R,S)-N-benzyl-N-(1-phenylethyl)-p-chlorobenzenesulfinamide 
• 1307296-50-9 (R,S)-N-benzyl-N-(1-phenylethyl)-p-fluorobenzenesulfinamide 
• 873-55-2 sodium benzenesulfonate 

Downstream Products

• 111698-33-0 (R)-methyl benzenesulfinate 
• 112425-42-0 (S)-methyl benzenesulfinate 
• 38235-77-7 (R)-N-benzyl-1-phenylethylamine 
• 13153-10-1 (S)-(-)-n-butyl phenyl sulfoxide 
• 1307296-52-1 (R,R)-N-benzyl-N-(1-phenylethyl)-p-toluenesulfinamide 
• 1307296-48-5 (R,S)-N-Benzyl-N-(1-phenylethyl)-p-toluenesulfinamide 
• 1307296-53-2 (R,R)-N-benzyl-N-(1-phenylethyl)-p-chlorobenzenesulfinamide 
• 1307296-49-6 (R,S)-N-benzyl-N-(1-phenylethyl)-p-chlorobenzenesulfinamide 
• 1307296-54-3 (R,R)-N-benzyl-N-(1-phenylethyl)-p-fluorobenzenesulfinamide 
• 1307296-50-9 (R,S)-N-benzyl-N-(1-phenylethyl)-p-fluorobenzenesulfinamide 

Relevant academic research and scientific papers

2-AMINO-N-(ARYLSULFINYL)-ACETAMIDE COMPOUNDS AS INHIBITORS OF BACTERIAL AMINOACYL-TRNA SYNTHETASE

The present invention pertains generally to the field of therapeutic compounds. More specifically the present invention pertains to certain 2-amino-N-(arylsulfinyl)- acetamide compounds that, inter alia, inhibit (e.g., selectively inhibit) bacterial amino

Practical and highly stereoselective method for the preparation of several chiral arylsulfinamides and arylsulfinates based on the spontaneous crystallization of diastereomerically pure N-benzyl-N-(1-phenylethyl)- arylsulfinamides

A novel and simple process for the preparation of enantiomerically pure (SS)-benzenesulfinamide (SS)-3a, (SS)-p- toluenesulfinamide (SS)-3b, (SS)-p-chloro- benzenesulfinamide (SS)-3c and (SS)-p- fluorobenzenesulfinamide (SS)-3d has been developed. The treatment of arylsulfinyl chlorides with (R)-N-benzyl-1-phenylethanamine in the presence of excess triethylamine gave diastereomeric mixtures of N-benzyl-N-(1-phenylethyl)- arylsulfinamides 1, which underwent spontaneous crystallization to furnish diastereomerically pure (R,SS)-N-benzyl-N-(1-phenylethyl)- arylsulfinamides (R,SS)-1a-1d in 28%, 29%, 27% and 31% yields, respectively. The diastereomerically pure compounds (R,SS)-1 were then converted into four enantiopure (RS)-methyl arylsulfinates (RS)-2, and finally into four enantiopure (SS)- arylsulfinamides (SS)-3 in good yields.