1309792-07-1Relevant academic research and scientific papers
Palladium-catalyzed cross-coupling of 1-aminoazoles with aryl chlorides: Application to the synthesis of unsymmetrical N,N'-diaryl-1-aminoindoles
Brachet, Etienne,Messaoudi, Samir,Peyrat, Jean-Franaois,Brion, Jean-Daniel,Alami, Mouad
, p. 2829 - 2839,11 (2012/12/12)
An efficient method for the selective mono-N-arylation of 1-aminoazoles to provide a range of N-aryl-1-aminoazoles in good yields is described. This process based on the use of tris(dibenzylideneacetone) dipalladium associated to Xphos as the catalyst sys
Palladium-catalyzed cross-coupling of 1-aminoazoles with aryl chlorides: Application to the synthesis of unsymmetrical N,N'-diaryl-1-aminoindoles
Brachet, Etienne,Messaoudi, Samir,Peyrat, Jean-Franaois,Brion, Jean-Daniel,Alami, Mouad
, p. 2829 - 2839 (2013/01/15)
An efficient method for the selective mono-N-arylation of 1-aminoazoles to provide a range of N-aryl-1-aminoazoles in good yields is described. This process based on the use of tris(dibenzylideneacetone) dipalladium associated to Xphos as the catalyst sys
Palladium-catalyzed selective N-(hetero)arylation or N,N′-di(hetero) arylation of 1-aminoindoles
Messaoudi, Samir,Brion, Jean-Daniel,Alami, Mouad
scheme or table, p. 2687 - 2691 (2011/06/19)
The selective synthesis of N-(hetero)aryl-1-aminoindoles 3 from the corresponding N-aminoindoles and (hetero)aryl halides using a catalyst combination of Pd2(dba)3 associated to Josiphos is described. By switching to Xantphos as the
