1310460-32-2

Upstream product

• 70-11-1 α-bromoacetophenone 
• 128-44-9 saccharin sodium salt 
• 15246-95-4 1,1-dioxo-2-(2-oxo-2-phenyl-ethyl)-1,2-dihydro-1λ⁶-benzo[d]isothiazol-3-one 
• 919467-55-3 ethyl 2-(3-benzoyl-4-hydroxy-1,1-dioxido-2H-benzo[e][1,2]thiazin-2-yl)acetate 
• 61018-80-2 (4-hydroxy-1,1-dioxo-1,2-dihydro-1λ⁶-benzo[e][1,2]thiazin-3-yl)-phenyl-methanone 

Downstream Products

• 1310459-61-0 2-(3-benzoyl-4-hydroxy-1,1-dioxido-2H-benzo[e][1,2]thiazin-2-yl)-N-(furan-2-ylmethyl)acetamide 
• 1310459-20-1 2-(3-benzoyl-4-hydroxy-1,1-dioxido-2H-benzo[e][1,2]thiazin-2-yl)-N-adamantylacetamide 
• 1310459-62-1 2-(3-benzoyl-4-hydroxy-1,1-dioxido-2H-benzo[e][1,2]thiazin-2-yl)-N-(4-(trifluoromethyl)benzyl)acetamide 
• 1310459-65-4 2-(3-benzoyl-4-hydroxy-1,1-dioxido-2H-benzo[e][1,2]thiazin-2-yl)-N-(1-(4-fluorophenyl)ethyl)acetamide 
• 1310459-66-5 2-(3-benzoyl-4-hydroxy-1,1-dioxido-2H-benzo[e][1,2]thiazin-2-yl)-N-(4-ethylbenzyl)acetamide 
• 1310459-15-4 2-(3-benzoyl-4-hydroxy-1,1-dioxido-2H-benzo[e][1,2]thiazin-2-yl)-N-[3-(trifluoromethyl)phenyl]acetamide 
• 1310459-33-6 2-(3-benzoyl-4-hydroxy-1,1-dioxido-2H-benzo[e][1,2]thiazin-2-yl)-N-cyclohexylacetamide 
• 1310460-27-5 2-(3-benzoyl-4-hydroxy-1,1-dioxido-2H-benzo[e][1,2]thiazin-2-yl)-N-(p-tolyl)acetamide 
• 1310459-48-3 2-(3-benzoyl-4-hydroxy-1,1-dioxido-2H-benzo[e][1,2]thiazin-2-yl)-N-ethylacetamide 
• 1310459-57-4 2-(3-benzoyl-4-hydroxy-1,1-dioxido-2H-benzo[e][1,2]thiazin-2-yl)-N-(4-(methoxy)benzyl)acetamide 
• 1310459-49-4 2-(3-benzoyl-4-hydroxy-1,1-dioxido-2H-benzo[e][1,2]thiazin-2-yl)-N,N-diethylacetamide 
• 1310459-13-2 2-(3-benzoyl-4-hydroxy-1,1-dioxido-2H-benzo[e][1,2]thiazin-2-yl)-N-phenylacetamide 
• 1310459-60-9 2-(3-benzoyl-4-hydroxy-1,1-dioxido-2H-benzo[e][1,2]thiazin-2-yl)-N-(m-tolyl)acetamide 
• 1310459-63-2 2-(3-benzoyl-4-hydroxy-1,1-dioxido-2H-benzo[e][1,2]thiazin-2-yl)-N-(4-fluorobenzyl)acetamide 

Relevant academic research and scientific papers

Identification of cyclicsulfonamide derivatives with an acetamide group as 11β-hydroxysteroid dehydrogenase 1 inhibitors

In the continuation of our 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD1) inhibitor research, cyclic sulfonamide derivatives with an acetamide group at the 2-position were synthesized and evaluated for their abilities to inhibit 11β-HSD1. Among this s