1315257-97-6Relevant articles and documents
Palladium-/copper-catalyzed regioselective amination and chloroamination of indoles
Liu, Xue-Yuan,Gao, Pin,Shen, Yong-Wen,Liang, Yong-Min
supporting information; experimental part, p. 4196 - 4199 (2011/10/04)
A palladium-/copper-catalyzed intermolecular C-H amination reaction of indoles has been developed. This reaction proceeds in good to excellent yields to produce a variety of 2-amino-substituted indoles and exhibits excellent regioselectivity at room temperature. Furthermore, chloroamination of indoles provides a simple method for the construction of C-N and C-Cl bonds in one step.