131604-75-6Relevant academic research and scientific papers
Distinct CCK-2 receptor conformations associated with β-arrestin-2 recruitment or phospholipase-C activation revealed by a biased antagonist
Magnan, Rémi,Escrieut, Chantal,Gigoux, Véronique,De, Kavita,Clerc, Pascal,Niu, Fan,Azema, Joelle,Masri, Bernard,Cordomi, Arnau,Baltas, Michel,Tikhonova, Irina G.,Fourmy, Daniel
supporting information, p. 2560 - 2573 (2013/03/29)
Seven-transmembrane receptors (7TMRs), also termed G protein-coupled receptors (GPCRs), form the largest class of cell surface membrane receptors, involving several hundred members in the human genome. Nearly 30% of marketed pharmacological agents target
2,4-DIOXO-5-PHENYL-2,3,4,5-TETRAHYDRO-1H-1,5-ENZODIAZEPINES
-
, (2008/06/13)
A compound in all possible isomeric forms and mixtures thereof of the formula STR1 wherein X and X' are individually selected from the group consisting of hydrogen, halogen, cyano,--NO 2,--CF 3 and alkyl and alkoxy of 1 to 8 carbon atoms, R is hydrogen or alkyl of 1 to 8 carbon atoms and Ar is selected from the group consisting of an unsubstituted or substituted aryl of 6 to 14 carbon atoms, an unsubstituted or substituted aromatic heterocyclic or a heterocyclic united with an unsubstituted or substituted aryl having cholecystokinine antagonistic activity.
