13202-07-8Relevant academic research and scientific papers
Antitumor and anti-Pneumocystis carinii activities of novel bisbenzamidines
Vanden Eynde, Jean Jacques,Mayence, Annie,Johnson, Melissa T.,Huang, Tien L.,Collins, Margaret S.,Rebholz, Sandra,Walzer, Peter D.,Cushion, Melanie T.,Donkor, Isaac O.
, p. 143 - 157 (2007/10/03)
Among a library of 17 bisbenzamidines connected with various linkers, compounds with a flexible pentanediamide (10) or hexanediamide (12) linker were the most potent derivatives against rat Pneumocystis carinii (IC50 values of 3 and 2 nM, respe
