133010-27-2Relevant academic research and scientific papers
A convenient synthesis of 1,3,4-thiadiazole and 1,3,4-oxadiazole based peptidomimetics employing diacylhydrazines derived from amino acids
Nagendra,Lamani, Ravi S.,Narendra,Sureshbabu, Vommina V.
body text, p. 6338 - 6341 (2011/01/04)
Synthesis of novel orthogonally protected 1,3,4-thiadiazole and 1,3,4-oxadiazole tethered dipeptide mimetics is described. Both the heterocycles are prepared via a set of diacylhydrazines derived from amino acids. 1,3,4-Thiadiazoles are synthesized by deh
Synthesis of Boc- and Z-protected amino acid fluorides employing DAST as a fluorinating agent
Suresh Babu,Gopi,Ananda
, p. 384 - 386 (2007/10/03)
DAST [(diethylamino)sulphur trifluoride] has been used as a fluorinating agent for the synthesis of Boc- and Z-protected amino acid fluorides. All the compounds made have been isolated as crystalline solids in good yield and purity.
tert-Butyloxycarbonyl and Benzyloxycarbonyl Amino Acid Fluorides. New, Stable Rapid-Acting Acylating Agents for Peptide Synthesis
Carpino, Louis A.,Mansour, El-Sayed M. E.,Sadat-Aalaee, Dean
, p. 2611 - 2614 (2007/10/02)
A new class of rapid-acting acylating agents, α-BOC and Z amino acid fluorides are obtained as stable, often crystalline, compounds by treatment of the protected amino acid cyanuric fluoride.
