134133-77-0Relevant articles and documents
Electrophilic γ-Lactone κ-Opioid Receptor Probes. Analogues of 2'-Hydroxy-2-tetrahydrofurfuryl-5,9-dimethyl-6,7-benzomorphan Diastereomers
Klein, Peter,Nelson, Wendel L.
, p. 2438 - 2444 (2007/10/02)
Benzomorphans with an electrophilic group in the nitrogen substituent were prepared as potentially irreversible ligands for the κ-opioid receptor.These were synthesized from products of the reaction of normetazocine with the enantiomers of 5-(iodomethyl)-