134362-19-9Relevant articles and documents
Convenient Approach to 2-Substituted (Thio)morpholin-3-ones from α-Diazoacetates via X-H Carbene Insertion – Lactamization Sequence
Solovyov, Igor,Dar'in, Dmitry,Krasavin, Mikhail
, p. 7432 - 7438 (2019)
Stepwise coupling of N-Boc-protected β-aminoethanols or β-mercaptoethylamines with various α-diazoacetates provides a new, unified approach to constructing (thio)morpholin-3-ones. The process involves a Rh2(esp)2-catalyzed X-H insert