1346523-92-9Relevant academic research and scientific papers
Exploiting the acylating nature of the imide-ugi intermediate: A straightforward synthesis of tetrahydro-1,4-benzodiazepin-2-ones
Mossetti, Riccardo,Saggiorato, Desiree,Tron, Gian Cesare
, p. 10258 - 10262 (2012/02/02)
We describe a simple and novel protocol for the synthesis of tetrahydro-1,4-benzodiazepin-2-ones with three points of diversity, exploiting the acylating properties of the recently rediscovered Ugi-imide. The final compounds can be easily prepared in thre
