134842-98-1Relevant articles and documents
Pyrazolo[1′,5′:1,6]pyrimido[4,5-d]pyridazin-4(3H)-ones as selective human A1 adenosine receptor ligands
Giovannoni, Maria Paola,Vergelli, Claudia,Cilibrizzi, Agostino,Crocetti, Letizia,Biancalani, Claudio,Graziano, Alessia,Piaz, Vittorio Dal,Loza, Maria Isabel,Cadavid, Maria Isabel,Díaz, José Luis,Gavald, Amadeu
scheme or table, p. 7890 - 7899 (2011/01/13)
A series of pyrazolo[1′,5′:1,6]pyrimido[4,5-d]pyridazin-4(3H)- ones was synthesized and tested in radioligand binding assays to determine their affinities for the human adenosine A1, A2A, A 2B and A3 receptors.